Orlistat

Orlistat (CAS 96829-58-2) is a potent, reversible inhibitor of gastrointestinal lipases, supplied as a white to off-white crystalline powder with 99% purity meeting USP specifications. It works by binding to the active site of pancreatic and gastric lipases, preventing the hydrolysis of dietary triglycerides into absorbable free fatty acids. This mechanism reduces fat absorption by approximately 30%, making it a key active ingredient in weight management formulations.

Our orlistat is produced under strict GMP conditions and is available in bulk quantities for pharmaceutical and nutraceutical manufacturers. Each batch is thoroughly tested to ensure compliance with USP standards, providing consistent quality for your formulations.

Synonyms: Tetrahydrolipstatin, THL, N-Formyl-L-leucine (1S,3S,7S,10S,13R,16R,17R)-1,3,7,10,13,16-hexamethyl-2,4,6,9,12,15-hexaoxo-17-(2-methylpropyl)-1,2,3,4,5,6,7,8,9,10,11,12,13,14,15,16-hexadecahydrocyclopenta[f][1]benzoxacyclotetradecin-16-yl ester, (2S,3S,5S,7S,10S,13S,16R,17R)-17-(2-methylpropyl)-2,3,5,7,10,13,16-hexamethyl-4,6,9,12,15-hexaoxo-1,17-dioxacyclotetradec-1-yl ester

Applications

• Weight management and anti-obesity pharmaceutical formulations (e.g., capsules, tablets)
• OTC dietary supplements for fat absorption control
• Clinical research and development for metabolic disorders
• Combination therapies with other weight-loss agents

Quality & Documentation

Every batch is tested for assay (HPLC ≥99%), loss on drying (≤0.5%), and heavy metals (≤10 ppm). Full COA, MSDS, and TDS are provided with each shipment. Stability data and regulatory support documents are available on request for qualification purposes.

Packaging & Supply

We supply orlistat in standard packaging of 1 kg, 5 kg, and 25 kg, with custom packing options available. In-stock items ship within 3-5 days; MOQ is 1 kg. For pricing, samples, and bulk orders, contact our sales team.

Request For Quote

• Our Address: 280 Main Street, Xian, Shaanxi, China
• LyvBio Co., Ltd. — Email: info@lyvbio.com