Amino Tadalafil

Synonyms

Amino Tadalafil, 6-Aminotadalafil, 6-amino-1,3-benzodioxole-5-carboxamide derivative, (6R,12aR)-6-amino-2,3,6,7,12,12a-hexahydropyrazino[1′,2′:1,6]pyrido[3,4-b]indole-1,4-dione

Amino Tadalafil is the amino-modified version of the well-known PDE5 inhibitor tadalafil. It’s not just an intermediate—it’s a versatile building block for researchers developing next-generation erectile dysfunction treatments and pulmonary hypertension therapies. The amino group opens up new conjugation possibilities, making it a valuable tool for prodrug design and targeted delivery.

For manufacturers, this means a reliable, high-purity compound that can be used in complex synthesis without worrying about impurities. We supply it as a white crystalline powder, with every batch rigorously tested to ensure consistency. Whether you need a few grams for R&D or kilograms for scale-up, we have flexible packaging options and can ship worldwide with full documentation.

Function

• PDE5 Inhibition: Retains the core pharmacophore of tadalafil, offering potent and selective inhibition of PDE5, which supports smooth muscle relaxation and increased blood flow.
• Chemical Intermediate: The primary amino group allows for easy derivatization, enabling the synthesis of novel analogs with improved pharmacokinetic profiles.

Source & Purity

• Source: Synthetic, produced under controlled conditions.
• Purity: ≥99% by HPLC, ensuring high batch-to-batch consistency.
• Appearance: White to off-white powder.

Documentation & Supply

• Documentation: COA, MSDS, TDS
• Lead time: 3-5 working days for in-stock items; custom quantities available upon request.
• Packaging: 10g, 100g, 1kg, or custom packaging to meet your needs.

Request For Quote

• Our Address: 280 Main Street, Xian, Shaanxi, China
• LyvBio Co., Ltd. — Email: info@lyvbio.com